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Introduction to Photostability
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Drug-Like Properties in Drug Discovery
| Type | Course |
|---|---|
| Language | English |
| Date |
April 5, 2008
to April 6, 2008 |
| Venue |
Sheraton at Woodbridge Place Hotel 515 US Highway 1 South Iselin, New Jersey 08830 US |
| Chemistry Specialties |
|
| Chemistry Techniques |
|
| Contact |
ACS 1155 Sixteenth Street, NW Washington, DC , 20036 US 1-800-227-5558 ext. 4508 202-872-6336 service@acs.org |
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This course is designed to increase your knowledge of drug-like properties, ADME and how to apply this information in medicinal chemistry for hit selection, lead optimization and development candidate selection and is designed for medicinal chemists and other discovery scientists who design, synthesize, and test new drug candidates, lead research teams, or measure and predict ADMET properties of compounds. Registrants will receive a copy of the text, Drug-Like Properties: Concepts, Structure Design and Methods: From ADME to Toxicology, as part of this course.
Key Topics
• Essentials of key pharmaceutical properties and practical real-world applications
• Successful structure modification strategies to improve drug-like properties and pharmacokinetics.
• Case studies on how med chemists enhance properties and PK through structure modification.
• The impact of drug properties on drug discovery chemistry, in vitro and in vivo biological testing, pharmacokinetics, and safety.
• Property assays: experimental design, measurement and interpretation.
• Which properties to optimize for improved pharmacokinetics performance.
Speakers
Edward H. Kerns is Associate Director of Chemical Technologies in Drug Discovery at Wyeth Research. He leads the pharmaceutical profiling group to provide property data for drug discovery compounds.
Li Di is Principal Research Scientist II in Chemical Technologies in Drug Discovery at Wyeth Research. She is the group leader for property profiling in Princeton and consults for teams on property optimization.
Cost
Note : The course fee includes all course materials, continental breakfast and lunch each day.
Member : $1,195
Academic Member : $597.50
Note: This discount is only available if you register by fax, mail or phone and mention this discount and may not be combined with any other offer.
Nonmember : $1,345
Early Registration : Register before January 14, 2008 for the Woodbridge Circuit and receive $100 off the standard member/nonmember fees.
Late Registration : Registrations after February 4, 2008 for the Woodbridge Circuit will be assessed a $100 administrative fee.
Group Rate : Five for Four! Register five people for one course, one person for five courses, or any combination in between and your fifth registration is free.
Note: This discount is only available if you register by fax, mail or phone and mention this discount and may not be combined with any other offer.